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PKC-theta inhibitor
CAS No. 736048-65-0
PKC-theta inhibitor( —— )
Catalog No. M20187 CAS No. 736048-65-0
PKC-theta inhibitor is PKC-θinhibitor with an?IC50?of 12 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 239 | In Stock |
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| 10MG | 381 | In Stock |
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| 100MG | Get Quote | In Stock |
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| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NamePKC-theta inhibitor
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NoteResearch use only, not for human use.
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Brief DescriptionPKC-theta inhibitor is PKC-θinhibitor with an?IC50?of 12 nM.
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DescriptionPKC-theta inhibitor is PKC-θinhibitor with an?IC50?of 12 nM.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayAngiogenesis
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TargetPKC
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RecptorPKCθ
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Research Area——
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Indication——
Chemical Information
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CAS Number736048-65-0
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Formula Weight454.4
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Molecular FormulaC20H25F3N6O3
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Purity>98% (HPLC)
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SolubilityDMSO:62.5 mg/mL?(137.53 mM)
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SMILESNCC1CCC(CNc2nc(NCc3ccccc3OC(F)(F)F)ncc2[N+]([O-])=O)CC1
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Chemical NameN4-((4-(aminomethyl)cyclohexyl)methyl)-5-nitro-N2-(2-(trifluoromethoxy)benzyl)pyrimidine-24-diamine
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Cywin CL et al. Discovery of potent and selective PKC-theta inhibitors. Bioorg Med Chem Lett. 2007 Jan 1;17(1):225-30.
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